Researcher interests: Peptides, synthesis, biology and conformation. Conversion of peptides into drugs. Tyrosine kinase inhibitors as antiproliferative drugs.
FACULTY / SCHOOL: Faculty of Science
DEPARTMENT: The Institute of Chemistry
Selected Publications
diffusion enhanced amide bond formation on a solid support (2019)|
Organic Process Research & Development|
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deciphering direct and indirect effects of neurokinin b and gnrh in the brain pituitary axis of tilapia (2019)|
Frontiers in Endocrinology|
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myristoylation confers oral bioavailability and improves the bioactivity of c myd 4 4 a cyclic peptide inhibitor of myd88 (2019)|
Molecular Pharmaceutics|
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molecular basis of neural memory definingthe engram (2018)|
Research in Medical & Engineering Sciences|
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development of a novel backbone cyclic peptide inhibitor of the innate immune tlr il1r signaling protein myd88 (2018)|
Scientific Reports|
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orally active peptides is there a magic bullet (2018)|
Angewandte Chemie|
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oral aktive peptide gibt es ein patentrezept (2018)|
Angewandte Chemie|
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enhancing the efficiency of the solid phase peptide synthesis spps process by high shear mixing (2018)|
Organic Process Research & Development|
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enhancing oral bioavailability of cyclic rgd hexa peptides by the lipophilic prodrug charge masking approach redirection of peptide intestinal permeability from paracellular to transcellular pathway (2018)|
Molecular Pharmaceutics|
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conversion of protein active regions into peptidomimetic therapeutic leads using backbone cyclization and cycloscan how to do it yourself (2018)|
Current Topics in Medicinal Chemistry|
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optimization of chemical processes by the hydrodynamic simulation method hsm (2018)|
ChemEngineering|
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overcoming the lack of oral availability of cyclic hexapeptides design of a selective and orally available ligand for the integrin αvβ3 (2017)|
Angewandte Chemie|
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frontispiece a tandem in situ peptide cyclization through trifluoroacetic acid cleavage (2014)|
Angewandte Chemie|
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a tandem in situ peptide cyclization through trifluoroacetic acid cleavage (2014)|
Angewandte Chemie|
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a comparative study of backbone versus side chain peptide cyclization application for hiv 1 integrase inhibitors (2012)|
Bioorganic & Medicinal Chemistry|
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